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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50197929(CHEMBL3954506)
Affinity DataIC50:  17nMAssay Description:Inhibition of human cathepsin K expressed in Pichia pastoris using Z-Phe-Arg-AMC as substrate after 30 mins by spectromicrofluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50197929(CHEMBL3954506)
Affinity DataIC50:  23nMAssay Description:Inhibition of human cathepsin L using Z-Phe-Arg-AMC as substrate after 30 mins by spectromicrofluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50197929(CHEMBL3954506)
Affinity DataIC50:  28nMAssay Description:Inhibition of human cathepsin S using Z-LR-AMC as substrate after 30 mins by spectromicrofluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50197929(CHEMBL3954506)
Affinity DataIC50:  79nMAssay Description:Inhibition of human cathepsin B using Z-Phe-Arg-AMC as substrate after 30 mins by spectromicrofluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed