Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCaspase-1(Homo sapiens (Human))
Basf Bioresearch

Curated by ChEMBL
LigandPNGBDBM50091570(3-[2-(2-Benzyloxycarbonylamino-3-methyl-butyrylami...)
Affinity DataIC50:  17nMAssay Description:Dissociation constant for inhibition of caspase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Homo sapiens (Human))
Basf Bioresearch

Curated by ChEMBL
LigandPNGBDBM50091570(3-[2-(2-Benzyloxycarbonylamino-3-methyl-butyrylami...)
Affinity DataKoff:  1.60E+5s-1Assay Description:Evaluated for kinetic dissociation constant (kon) for the inhibition of caspase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed