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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetG protein-coupled receptor 119(Macaca fascicularis)
Amgen

Curated by ChEMBL
LigandPNGBDBM50445481(CHEMBL3104879)
Affinity DataEC50:  73nMAssay Description:Agonist activity at cynomolgus monkey GPR119 assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Mus musculus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50445481(CHEMBL3104879)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at mouse GPR119 assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50445481(CHEMBL3104879)
Affinity DataEC50:  2.05E+3nMAssay Description:Agonist activity at rat GPR119 assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50445481(CHEMBL3104879)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as cAMP accumulation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed