Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL

LigandBDBM50518986(CHEMBL4584173)Copy SMILESCopy InChI

Affinity DataIC50:  6.5nMAssay Description:Antagonist activity at beta2 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL

LigandBDBM50518986(CHEMBL4584173)Copy SMILESCopy InChI

Affinity DataIC50:  28nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI