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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Gamma-aminobutyric acid type B receptor subunit 1/2
(Homo sapiens (Human))
Beijing Institute Of Biotechnology
Curated by
ChEMBL
Ligand
BDBM50550633
(CHEMBL4763515)
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Affinity Data
IC50: 0.200nM
Assay Description:
Activation of human GABAB1/GABAB2 expressed in HEK293 cells co-transfected with rat CaV2.2 channel assessed as reduction in CaV2.2-mediated peak-curr...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Nicotinic acetylcholine receptor alpha9/alpha10
(RAT)
Beijing Institute Of Biotechnology
Curated by
ChEMBL
Ligand
BDBM50550633
(CHEMBL4763515)
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Copy InChI
Affinity Data
IC50: 875nM
Assay Description:
Inhibition of rat alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -80 mV holding potential ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuronal acetylcholine receptor; alpha9/alpha10
(Homo sapiens (Human))
Beijing Institute Of Biotechnology
Curated by
ChEMBL
Ligand
BDBM50550633
(CHEMBL4763515)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.93E+3nM
Assay Description:
Inhibition of human alpha9alpha10 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -80 mV holding potentia...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
KEGG
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI