Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 82 hits in this display
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
IC50: 3.10nMAssay Description:Dopaminergic activity assessed in vitro for displacement of [3H]apomorphine from specific binding sites on rat striatal membranesMore data for this Ligand-Target Pair
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
IC50: 18nMAssay Description:Inhibitory activity against rat striatal synaptosomes Dihydrodipicolinate reductase using 10 uM qBH2 and 50 uM NADH assaysMore data for this Ligand-Target Pair
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
IC50: 41nMAssay Description:Alpha-2 adrenergic receptor activity assessed in vitro for displacement of [3H]clonidine from specific binding sites on rat striatal membranesMore data for this Ligand-Target Pair
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
IC50: 70nMAssay Description:In vitro binding affinity towards dopamine receptor was determined in rat striatal membrane using [3H]spiroperidol as the radioligandMore data for this Ligand-Target Pair
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
IC50: 7.90E+3nMAssay Description:Inhibition of alpha-synuclein fibril formation (unknown origin) incubated for 6 days by thioflavin S based fluorescence assayMore data for this Ligand-Target Pair
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50028421(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
BDBM50017543((6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,...)
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