Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]MCH from human recombinant MCH1R expressed on CHOK1 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50:  20nMAssay Description:Antagonistic activity against MCH1R expressed on CHOK1 cells assessed as intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human ERG potassium channel 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of histamine H2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of adenosine receptor A2AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of mu-type opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of delta-type opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50301095(4-(4-fluorobenzyloxy)-1-(4-((propylamino)methyl)ph...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of kappa-type opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed