Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 363 hits in this display
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant Haspin (471 to end residues) using RARTLSFAEPG as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human CDKL2 in presence of 10 uM ATP by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human HCK recombinant (230 to 497 residues) using KVEKIGEGTYGVV as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HIPK1 (158 to 555 residues) using myelin basic protein as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HIPK3 (161 to 562 residues) using myelin basic protein as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human mTOR measured after 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human DNA-PK using GST-cMyc-p53 as substrate incubated for 40 mins by fluorescence assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant activated HCK (230 to 497 residues) using GGMEDIYFEFMGG as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant full length HIPK4 using RRRFRPASPLRGP as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HPK1 (1 to 346 residues) using myelin basic protein as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HRI (140 to end residues) using RSRSRSRSRSRSR as substrate after 120 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human CDK14/cyclinY in presence of [gamma-33ATP] by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of recombinant full length human CDKL4 in presence of [gamma-33ATP] by radiometric scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Inhibition of human GSK-3beta H350L mutant (2 to end residues) using YRRAAVPPSPSLSR as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
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