Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM50061008
(CHEMBL3393556 | US9732087, 96)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1nM
Assay Description:
Cell pellets from SK-N-MC cells stably or transiently transfected with human H4 receptor (NCBI accession No. AF312230) were used for the binding assa...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM50061008
(CHEMBL3393556 | US9732087, 96)
Copy SMILES
Copy InChI
Affinity Data
Ki: 8nM
Assay Description:
Displacement of [3H]histamine from human recombinant histamine H4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Ligand
BDBM50061008
(CHEMBL3393556 | US9732087, 96)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.00E+3nM
Assay Description:
Agonist activity at human recombinant histamine H4 receptor expressed in SK-N-MC cells assessed as effect on forskolin-stimulated cAMP-mediated repor...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI