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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
136
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 0.100nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.158nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 0.240nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.25nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human cloned 5-HT1A receptor expressed in CHO cells after 60 mins by liquid scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.330nM
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.331nM
Assay Description:
Displacement [3H]8-OH-DPAT of human cloned 5HT1A receptor expressed in human HeLa cells by rapid filtration technique
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.331nM
Assay Description:
Displacement of [3H]-OH-DPAT from human recombinant 5HT1A receptor expressed in HeLa cells after 30 mins by liquid scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.331nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human recombinant 5-HT1A receptor expressed in human HeLa cells incubated for 30 mins by radioligand competition ...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.331nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human cloned 5HT-1AR transfected in HeLa cells incubated for 30 mins by liquid scintillation counter
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Target
5-hydroxytryptamine receptor 1D
(Mus musculus (Mouse))
National Institutes Of Health
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 0.340nM
Assay Description:
Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]-GTP-gammaS, binding (Experi...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.390nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 EBNA cells after 2 hrs by liquid scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.390nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptor expressed in HEK293 EBNA cells after 1 hr by liquid scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 0.5nM
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 0.501nM
Assay Description:
Compound was tested for inhibition constant against 5-hydroxytryptamine 1A receptor in rat frontal cortex membranes.
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.501nM
Assay Description:
Binding affinity at human 5-hydroxytryptamine 1A receptor by inhibition of [3H]8-OH-DPAT binding in Chinese hamster ovary cell line
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.590nM
Assay Description:
Compound was tested in vitro for the inhibition of [3H]- 8-OH-DPAT binding to cloned cell line containing human 5-hydroxytryptamine 1A receptor
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.600nM
Assay Description:
Displacement of [3H]8-OH-DPAT from 5HT1A receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.600nM
Assay Description:
Inhibitory constant was determined against 5-hydroxytryptamine 1A receptor using 1.2 nM [3H]8-OH-DPAT
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.794nM
Assay Description:
Displacement of [3H]WAY100635 from human recombinant 5HT1A receptor
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.840nM
Assay Description:
Inhibition of binding of [125I]8-OH-PIPAT ligand to 5-hydroxytryptamine 1A receptor of rat hippocampal homogenates
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.900nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.900nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.900nM
Assay Description:
Displacement of 8-OH-DPAT from human 5-hydroxytryptamine 1A receptor expressed in chinese hamster ovary cells
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.900nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in CHO cells
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 0.960nM
Assay Description:
Binding affinity against human 5-hydroxytryptamine 1A receptor in CHO cells labeled with [3H]-8-OH-DPAT radioligand
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.960nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptor expressed in CHO cells
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.960nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO cells
More data for this Ligand-Target Pair
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Target
5-hydroxytryptamine receptor 1D
(Mus musculus (Mouse))
National Institutes Of Health
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 1.10nM
Assay Description:
Receptor-linked G protein activation at 5-hydroxytryptamine receptor was determined by measuring the stimulation of [35S]GTP-gamma-S, binding (Experi...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 2.20nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human recombinant 5HT1A receptor expressed in HEK293 cells after 120 mins
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 2.20nM
Assay Description:
Inhibition of 5HT1A receptor
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 4.57nM
Assay Description:
Displacement [3H]prazosin of human recombinant Alpha-1D adrenergic receptor expressed in CHO cells by rapid filtration technique
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 4.57nM
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4.57nM
Assay Description:
Displacement of [3H]prazosin from human recombinant Alpha-1D adrenoreceptor expressed in CHO cells after 30 mins by liquid scintillation counting
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: 4.60nM
Assay Description:
Displacement of [3H]Prazosin from human recombinant alpha 1D adrenergic receptor expressed in CHO cells incubated for 30 mins by radioligand competit...
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 4.60nM
Assay Description:
Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...
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Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 5nM
Assay Description:
Displacement of [3H]prazosin from Alpha-1D receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 16nM
Assay Description:
Inhibition of dopamine D4 receptor
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 16nM
Assay Description:
Displacement of [3H]N-methylspiperone from dopamine D4 receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 16.4nM
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 18.6nM
Assay Description:
Displacement of [3H]prazosin from human recombinant alpha1A adrenoceptor expressed in CHO cells after 30 mins by liquid scintillation counting
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 18.6nM
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 18.6nM
Assay Description:
Displacement [3H]prazosin of human recombinant alpha1A adrenergic receptor expressed in CHO cells by rapid filtration technique
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 19nM
Assay Description:
Displacement of [3H]Prazosin from human recombinant alpha 1A adrenergic receptor expressed in CHO cells incubated for 30 mins by radioligand competit...
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 19nM
Assay Description:
Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1A expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 19.9nM
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 20nM
Assay Description:
Inhibition of adrenergic alpha1A receptor
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Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 20nM
Assay Description:
Displacement of [3H]prazosin from alpha1A receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 24nM
Assay Description:
Displacement of [3H]LSD from 5HT2B receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
5-hydroxytryptamine receptor 2B
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 24nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 24nM
Assay Description:
Inhibition of 5HT1B receptor
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Target
Alpha-1A adrenergic receptor
(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 45nM
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 52nM
Assay Description:
Displacement of [3H]-YM-09151-2 from human cloned D4 receptor expressed in Sf9 cells after 60 mins by liquid scintillation counting
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 66nM
Assay Description:
Displacement of [3H]Prazosin from human recombinant alpha 1B adrenergic receptor expressed in CHO cells incubated for 30 mins by radioligand competit...
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 66nM
Assay Description:
Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1B expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 66.1nM
Assay Description:
Displacement [3H]prazosin of human recombinant Alpha-1B adrenergic receptor expressed in CHO cells by rapid filtration technique
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 66.1nM
Assay Description:
Displacement of [3H]prazosin from human recombinant alpha1B adrenoceptor expressed in CHO cells after 30 mins by liquid scintillation counting
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Target
D(3) dopamine receptor
(Homo sapiens (Human))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 67nM
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Target
D(2) dopamine receptor
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 78nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 79nM
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Target
Alpha-1A adrenergic receptor
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 120nM
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Target
5-hydroxytryptamine receptor 2C isoform A
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 282nM
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 322nM
Assay Description:
Displacement of [3H]prazosin from Alpha-1B receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 322nM
Assay Description:
Inhibition of adrenergic alpha1B receptor
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 322nM
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Target
D(2) dopamine receptor
(Rattus norvegicus (rat))
Universit&Aagrove
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 347nM
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Target
D(3) dopamine receptor
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 370nM
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Target
D(3) dopamine receptor
(Rattus norvegicus (Rat))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 370nM
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Target
Kappa-type opioid receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 412nM
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Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 661nM
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Target
D(2) dopamine receptor
(Homo sapiens (Human))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 940nM
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Target
Alpha-2C adrenergic receptor
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 1.00E+3nM
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Target
D(1A) dopamine receptor
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 1.00E+3nM
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Target
Beta-2 adrenergic receptor
(Rattus norvegicus)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 1.00E+3nM
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Target
Muscarinic acetylcholine receptor M2
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 1.00E+3nM
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Target
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+3nM
Assay Description:
Binding affinity against serotonin transporter in rat cortical tissues using radioligand [3H]-paroxetine
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Target
5-hydroxytryptamine receptor 2A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 1.10E+3nM
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Target
Alpha-2C adrenergic receptor
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 1.26E+3nM
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Target
5-hydroxytryptamine receptor 2A
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 1.91E+3nM
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Target
5-hydroxytryptamine receptor 1D
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 2.45E+3nM
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Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 2.57E+3nM
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Target
Galanin peptides
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 2.60E+3nM
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Target
5-hydroxytryptamine receptor 2A
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: 6.26E+3nM
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Target
5-hydroxytryptamine receptor 1B
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 8.31E+3nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: 1.00E+4nM
Assay Description:
Inhibition of 5HT7 receptor
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Displacement of [3H]LSD from 5HT7 receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Displacement of [3H]GR127543 from 5HT1D receptor expressed in HEK293 EBNA cells by radioligand binding assay
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Target
5-hydroxytryptamine receptor 3A
(pigeon)
Cns-Pharmacology
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Gamma-aminobutyric acid receptor subunit alpha-1
(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Gamma-aminobutyric acid receptor subunit alpha-1
(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Ki: >1.00E+4nM
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Target
Glutamate receptor 3
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Histamine H1 receptor
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Histamine H2 receptor
(Cavia porcellus (domestic guinea pig))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Nicotinic acetylcholine receptor
(RAT)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1B
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1D
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1E
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 2C
(Rattus norvegicus (Rat))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 5A
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 6
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 7
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Alpha-2B adrenergic receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Beta-1 adrenergic receptor
(Rattus norvegicus (Rat))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
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Target
Beta-2 adrenergic receptor
(Rattus norvegicus)
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
Muscarinic acetylcholine receptor M5
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
Ki: >1.00E+4nM
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Target
D(1A) dopamine receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
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Target
D(1B) dopamine receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Gamma-aminobutyric acid receptor subunit alpha-1
(Rattus norvegicus (Rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Histamine H1 receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Histamine H2 receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Histamine H3 receptor
(GUINEA PIG)
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Histamine H4 receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Mu-type opioid receptor
(Homo sapiens (Human))
Purdue University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Ki: >1.00E+4nM
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 0.370nM
Assay Description:
In vitro affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT in rat hippocampus
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 0.910nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptor expressed in HEK293 EBNA cells after 1 hr by liquid scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 0.910nM
Assay Description:
Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 EBNA cells after 2 hrs by liquid scintillation counting
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 2.10nM
Assay Description:
Antagonist activity at human recombinant 5-HT1A receptor assessed as inhibition of 8-OH-DPAT-induced response by cellular dielectric spectroscopy
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 2.20nM
Assay Description:
Inhibitory activity against 5-hydroxytryptamine 1A receptor of rat hippocampal homogenates
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 2.20nM
Assay Description:
In vitro binding affinity to 5-hydroxytryptamine 1A receptor using [125I](R)-(+)-trans-8-OH-PIPAT as radioligand in rat hippocampal homogenate
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 2.80nM
Assay Description:
Antagonist activity at human 5HT1A receptor expressed in CHO-K1 cells assessed as inhibition of 5HT-induced calcium flux incubated for 60 mins at 37 ...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 4.04nM
Assay Description:
Activity at human cloned 5HT1A receptor expressed in CHO cells assessed as blockade of 5-HT-stimulated [35S]GTPgammaS binding
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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IC50: 4.20nM
Assay Description:
Displacement of [3H]-8-OH-DPAT from Sprague-Dawley rat hippocampal membrane 5HT1A receptor
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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IC50: 4.90nM
Assay Description:
Antagonist activity against human recombinant 5-HT1A receptor expressed in CHOK1 cells assessed as reduction in serotonin-induced increase in intrace...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 7.06nM
Assay Description:
Agonist activity at human 5HT1A receptor expressed in CHO cells by inhibition of 8-OH-DPAT-induced decrease in forskolin-stimulated cAMP production
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 7.10nM
Assay Description:
Antagonist activity at human 5HT1A receptor expressed in CHO cells assessed as blockade of 8-OH-DPAT-induced inhibition of forskolin-stimulated incre...
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
IC50: 8.40nM
Assay Description:
In vitro inhibition of 8-OH-DPAT-induced [35S]GTP-gamma-S, binding to 5-HT1A receptor/G protein complex in CHO cells
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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IC50: 11nM
Assay Description:
Antagonist activity at serotonin 5-HT1A receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of serotonin-induced calcium flux ...
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Target
Sodium-dependent serotonin transporter
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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IC50: >4.50E+3nM
Assay Description:
Inhibition concentration against [3H]-5-HT uptake by human serotonin transporter in JAR cells
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5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
EC50: 7.10nM
Assay Description:
Effective concentration against human 5-hydroxytryptamine 1A receptor using cAMP as radioligand in CHO cells
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Target
5-hydroxytryptamine receptor 1A
(Rattus norvegicus (rat))
Preclinical R & D, Astra Arcus
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Kd: 0.100nM
Assay Description:
In vitro binding affinity for 5-hydroxytryptamine 1A receptor was determined by measuring specific inhibition of [125I]-binding to rat hippocampal me...
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Kd: 0.200nM
Assay Description:
Binding affinity to 5-HT1A receptor (unknown origin) assessed as dissociation constant
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Target
D(4) dopamine receptor
(Homo sapiens (Human))
Vu University Medical Center
Curated by
ChEMBL
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
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Affinity Data
Kd: 2.40nM
Assay Description:
Binding affinity to D4 receptor (unknown origin) assessed as dissociation constant
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Target
5-hydroxytryptamine receptor 1A
(Homo sapiens (Human))
Sorbonne University
Curated by
PDSP K
i
Database
Ligand
BDBM86708
(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Copy SMILES
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Affinity Data
EC50: 7.10nM
Assay Description:
Effective concentration against binding of radioligand [35]GTPgammaS in CHO cells expressing human 5-hydroxytryptamine 1A receptor
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