Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 11 hits in this display
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
Ki: 2.60nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
Ki: 27nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
Prothrombin(Homo sapiens (Human))University of British Columbia
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
Ki: 9.27E+3nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
Ki: >1.00E+4nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
Furin(Homo sapiens (Human))University of British Columbia
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
Ki: >1.00E+4nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
IC50: 1.90nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
Hemagglutinin(Influenza A virus (strain A/X-31 H3N2))SociÉTÉ
US Patent
BDBM525152(Ms-QFR-kbt | N-0385 | US10988505, Example 2)
EC50: 9.33nMAssay Description:The ability of the tested compound to block influenza virus replication (PR8 and X31) in Calu-3 human bronchial epithelial cells was evaluated as des...More data for this Ligand-Target Pair