Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Transmembrane protease serine 6' and Ligand = 'BDBM525152'
TargetTransmembrane protease serine 6(Human)
University of British Columbia

LigandChemical structure of BindingDB Monomer ID 525152BDBM525152(US10988505, Example 2 | N-0385 | Ms-QFR-kbt)
Affinity DataKi:  2.60nMAssay Description:Vero E6 cells were transfected with mock (pcDNA3.1), TMPRSS2 (pcDNA3.1/TMPRSS2 Uniprot: O15393-1), or TMPRSS2-S441A (pcDNA3.1/TMPRSS2-S441A) using Li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetTransmembrane protease serine 6(Human)
University of British Columbia

LigandChemical structure of BindingDB Monomer ID 525152BDBM525152(US10988505, Example 2 | N-0385 | Ms-QFR-kbt)
Affinity DataKi:  2.63nMAssay Description:Enzymatic assays and Ki determination were performed at room temperature in an assay buffer containing 50 mM Tris-HCl, 150 mM NaCl and 500 μg/mL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details
US Patent