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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Nottingham

LigandPNGBDBM25765(Bupranolol | KL 255 | Ophtorenin | tert-butyl[3-(2...)
Affinity DataKd:  3.10nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University of Nottingham

LigandPNGBDBM25765(Bupranolol | KL 255 | Ophtorenin | tert-butyl[3-(2...)
Affinity DataKd:  91nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Nottingham

LigandPNGBDBM25765(Bupranolol | KL 255 | Ophtorenin | tert-butyl[3-(2...)
Affinity DataKd:  0.140nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank