Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL

LigandBDBM50516230(CHEMBL4532885)Copy SMILESCopy InChI

Affinity DataIC50:  763nMAssay Description:Inhibition of human beta5 20S immunoproteasome using Ac-ANW-AMC as substrateMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProteasome subunit beta type-5(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL

LigandBDBM50516230(CHEMBL4532885)Copy SMILESCopy InChI

Affinity DataIC50:  3.71E+4nMAssay Description:Inhibition of human beta5 20S constitutive proteasome using suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI