Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  1.84E+4nMAssay Description:Activation of recombinant human TREK1 G275C mutant expressed in HEK293T cells assessed as increase in K+ current amplitude in presence of MTSET by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  1.28E+4nMAssay Description:Activation of recombinant human TREK1 expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clamp electrophys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTREK-2 two-pore-domain K+ channel(Mus musculus)
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  1.13E+4nMAssay Description:Activation of recombinant mouse TREK2 expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clamp electrophys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  7.57E+3nMAssay Description:Activation of recombinant human TREK1 T156A mutant expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  3.91E+3nMAssay Description:Activation of recombinant human TREK1 W290A mutant expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  1.52E+4nMAssay Description:Activation of recombinant human TREK1 G275C mutant expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 4(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  1.53E+4nMAssay Description:Activation of recombinant human TRAAK expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clamp electrophys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  2.24E+4nMAssay Description:Activation of recombinant human TREK1 F149A mutant expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium channel subfamily K member 2(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50514764(CHEMBL4552751)
Affinity DataEC50:  7.98E+3nMAssay Description:Activation of recombinant human TREK1 I293A mutant expressed in HEK293T cells assessed as increase in K+ current amplitude by whole cell voltage clam...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed