Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM313774(US10167292, Example 8)
BDBM313774(US10167292, Example 8)
BDBM313774(US10167292, Example 8)
BDBM313774(US10167292, Example 8)
BDBM313774(US10167292, Example 8)
BDBM313774(US10167292, Example 8)
BDBM313774(US10167292, Example 8)
IC50: <100nMAssay Description:BRD binding and inhibition was assessed by measuring the interaction of biotinylated acetyl-histone H4 peptide (Anaspec #64989) with the BRD target p...More data for this Ligand-Target Pair
BDBM313774(US10167292, Example 8)
IC50: <100nMAssay Description:BRD binding and inhibition was assessed by measuring the interaction of biotinylated acetyl-histone H4 peptide (Anaspec #64989) with the BRD target p...More data for this Ligand-Target Pair
BDBM313774(US10167292, Example 8)
IC50: <100nMAssay Description:BRD binding and inhibition was assessed by measuring the interaction of biotinylated acetyl-histone H4 peptide (Anaspec #64989) with the BRD target p...More data for this Ligand-Target Pair
BDBM313774(US10167292, Example 8)
IC50: <100nMAssay Description:BRD binding and inhibition was assessed by measuring the interaction of biotinylated acetyl-histone H4 peptide (Anaspec #64989) with the BRD target p...More data for this Ligand-Target Pair
BDBM313774(US10167292, Example 8)
Kon: 0.130M-1s-1Assay Description:Binding affinity to His-tagged human Brd2 bromodomain 1 (1 to 473 residues) assessed as dissociation rate constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
BDBM313774(US10167292, Example 8)
Kon: 0.0390M-1s-1Assay Description:Binding affinity to His-tagged human Brd2 bromodomain 2 (1 to 473 residues) assessed as dissociation rate constant by surface plasmon resonance assayMore data for this Ligand-Target Pair