Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetGlycine receptor subunit alpha-1(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  1.07nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  11.5nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]granisectron from 5HT3 receptor in Wistar rat forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  33.9nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  70.8nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  126nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(RAT)
Hungarian Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Affinity DataIC50:  135nMAssay Description:Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed