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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Glycine receptor subunit alpha-1
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
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Affinity Data
IC50: 1.07nM
Assay Description:
Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Glycine receptor subunit alpha-1
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 11.5nM
Assay Description:
Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometry
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 3A
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
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Affinity Data
IC50: 25nM
Assay Description:
Displacement of [3H]granisectron from 5HT3 receptor in Wistar rat forebrain
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycine receptor subunit alpha-1
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 33.9nM
Assay Description:
Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometry
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycine receptor subunit alpha-1
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 70.8nM
Assay Description:
Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycine receptor subunit alpha-1
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 126nM
Assay Description:
Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometry
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glycine receptor subunit alpha-1
(RAT)
Hungarian Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50304335
(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 135nM
Assay Description:
Displacement of [3H]strychnine from GlyR low affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI