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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetCathepsin S(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50463221(CHEMBL4251253)
Affinity DataKi:  2nMAssay Description:Inhibition of human cathepsin S using Z-LR-AMC as substrate after 30 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50463221(CHEMBL4251253)
Affinity DataKi:  700nMAssay Description:Inhibition of human cathepsin K using Z-Phe-Arg-AMC as substrate after 30 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50463221(CHEMBL4251253)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibition of human cathepsin B using Z-Phe-Arg-AMC as substrate after 30 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50463221(CHEMBL4251253)
Affinity DataIC50:  3nMAssay Description:Inhibition of human cathepsin S using Z-LR-AMC as substrate after 30 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50463221(CHEMBL4251253)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human cathepsin K using Z-Phe-Arg-AMC as substrate after 30 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50463221(CHEMBL4251253)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human cathepsin B using Z-Phe-Arg-AMC as substrate after 30 mins by spectrofluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed