Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 84 hits in this display
IC50: >1.00E+4nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha 1A adrenoceptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]WIN55212-2 from recombinant human CB2 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [125I](+/-)DOI from recombinant human 5HT2A receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]nitrendipine from rat brain Cav1.2 dihydropyridine site after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]CGS21680 from recombinant human adenosine A2A receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]RX 821002 from recombinant human alpha 2A adrenoceptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP12177 from recombinant human beta2 adrenergic receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]7-OH-DPAT from recombinant human D2s receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [125I]endothelin-1 from recombinant human ETA receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]pirenzepine from recombinant human M1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [125I](+/-)DOI from recombinant human 5HT2B receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]nisoxetine from recombinant human norepinephrine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Activity at recombinant human LCK using Ulight-Poly GAT[EAY(1:1:1)]n as substrate measured after 10 mins by LANCE assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Activity at human recombinant COX1 using arachidonic acid as substrate measured after 3 mins by ADHP reagent based fluorescence assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Activity at human recombinant COX2 using arachidonic acid as substrate measured after 5 mins by ADHP reagent based fluorescence assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Activity at human recombinant ACHE using acetylthiocholine as substrate measured after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Activity at human recombinant PDE3A using [3H]cAMP as substrate measured after 15 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Activity at human recombinant PDE4D2 using [3H]cAMP as substrate measured after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP12177 from recombinant human beta1 adrenergic receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [125I]CCK-8s from recombinant human CCK1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]BRL43694 from recombinant human 5HT3 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]BTCP from recombinant human dopamine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]cytisine from recombinant human alpha4beta2 nAChR after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]pyrilamine from recombinant human H1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
IC50: >1.00E+4nMAssay Description:Displacement of [3H]imipramine from recombinant human serotonin transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [125I]endothelin-1 from recombinant human ETA receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]CGS21680 from recombinant human adenosine A2A receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]RX 821002 from recombinant human alpha 2A adrenoceptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP12177 from recombinant human beta2 adrenergic receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [125I]CCK-8s from recombinant human CCK1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]7-OH-DPAT from recombinant human D2s receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]BTCP from recombinant human dopamine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]cytisine from recombinant human alpha4beta2 nAChR after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]BRL43694 from recombinant human 5HT3 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Activity at human recombinant COX1 using arachidonic acid as substrate measured after 3 mins by ADHP reagent based fluorescence assayMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Activity at human recombinant PDE4D2 using [3H]cAMP as substrate measured after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [125I](+/-)DOI from recombinant human 5HT2B receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Activity at recombinant human LCK using Ulight-Poly GAT[EAY(1:1:1)]n as substrate measured after 10 mins by LANCE assayMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]imipramine from recombinant human serotonin transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Activity at human recombinant COX2 using arachidonic acid as substrate measured after 5 mins by ADHP reagent based fluorescence assayMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Activity at human recombinant ACHE using acetylthiocholine as substrate measured after 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Activity at human recombinant PDE3A using [3H]cAMP as substrate measured after 15 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha 1A adrenoceptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H](-)CGP12177 from recombinant human beta1 adrenergic receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]WIN55212-2 from recombinant human CB2 receptor after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]pyrilamine from recombinant human H1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]pirenzepine from recombinant human M1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [125I](+/-)DOI from recombinant human 5HT2A receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]nitrendipine from rat brain Cav1.2 dihydropyridine site after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
EC50: >1.00E+4nMAssay Description:Displacement of [3H]nisoxetine from recombinant human norepinephrine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
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