Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 20 hits in this display
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
IC50: 937nMAssay Description:Inhibition of recombinant full length C-terminal His-tagged human TDO expressed in Escherichia coli using L-Trp as substrate after 30 minsMore data for this Ligand-Target Pair
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)
BDBM48009(8-fluoranylindolo[2,1-b]quinazoline-6,12-dione | 8...)