Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 14 hits in this display
Ki: >4.00E+5nMAssay Description:Binding affinity to recombinant human BRD2 BD1 (72-205 residues) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ki: >4.00E+5nMAssay Description:Binding affinity to recombinant human BRD2 BD2 (349-460 residues) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ki: >4.00E+5nMAssay Description:Binding affinity to recombinant human BRD3 BD1 (24-144 residues) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ki: >4.00E+5nMAssay Description:Binding affinity to recombinant human BRD3 BD2 (306-417 residues) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair