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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Histamine H3 receptor
(Rattus norvegicus (rat))
Hokkaido University
Curated by
ChEMBL
Ligand
BDBM50127604
(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
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Affinity Data
Ki: 2.5nM
Assay Description:
Affinity against rat Histamine H3 receptor using [3H]-N-alpha-methyl histamine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Histamine H2 receptor
(Homo sapiens (Human))
Hokkaido University
Curated by
ChEMBL
Ligand
BDBM50127604
(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
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Affinity Data
EC50: >0.000100nM
Assay Description:
Inhibition of human Histamine H2 receptor using [3H]-tiotidine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Homo sapiens (Human))
Hokkaido University
Curated by
ChEMBL
Ligand
BDBM50127604
(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 96nM
Assay Description:
Inhibition of human Histamine H3 receptor using [3H]-N-alpha-methyl histamine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Hokkaido University
Curated by
ChEMBL
Ligand
BDBM50127604
(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >0.000100nM
Assay Description:
Inhibition of human Histamine H4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H1 receptor
(Homo sapiens (Human))
Hokkaido University
Curated by
ChEMBL
Ligand
BDBM50127604
(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >0.000100nM
Assay Description:
Inhibition of human Histamine H1 receptor using [3H]-pyrilamine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI