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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Aminopeptidase N
(Sus scrofa (Pig))
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
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Affinity Data
Ki: 0.0600nM
Assay Description:
Inhibition of porcine kidney APN using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysis
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aminopeptidase N
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
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Affinity Data
Ki: 0.0600nM
Assay Description:
Inhibition of human APN
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aminopeptidase N
(Sus scrofa (Pig))
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.0600nM
Assay Description:
Inhibition of pig APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectriphotometric analysis
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aminopeptidase N
(Mus musculus)
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
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Affinity Data
Ki: 0.200nM
Assay Description:
Inhibition of mouse APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectriphotometric analysis
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aminopeptidase N
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.350nM
Assay Description:
Inhibition of human APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectriphotometric analysis
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bacterial leucyl aminopeptidase
(Vibrio proteolyticus)
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
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Affinity Data
Ki: 3.90E+4nM
Assay Description:
Inhibition of Aeromonas proteolytica aminopeptidase using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cytosol aminopeptidase
(Bos taurus (bovine))
Universit£
Curated by
ChEMBL
Ligand
BDBM50353018
(CHEMBL1821980 | CHEMBL1852660)
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Copy InChI
Affinity Data
Ki: 7.00E+4nM
Assay Description:
Inhibition of bovine kidney cytosolic leucine aminopeptidase using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI