Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 25 hits in this display
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
IC50: 7.44E+3nMAssay Description:The inhibition of human CYP2A6-mediated 7-hydroxy coumarin formation was evaluated in the presence of 95 selected test compounds in a standard assay ...More data for this Ligand-Target Pair
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
IC50: 5.22E+4nMpH: 7.5Assay Description:To gain insight into the selectivity of the synthetic compounds for inhibition of other CYPs, we examined the major CYPs present in human liver. Prio...More data for this Ligand-Target Pair
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
IC50: 5.70E+4nMAssay Description:To gain insight into the selectivity of the synthetic compounds, nicotine, nicotine related alkaloids and nicotine metabolites for inhibition of othe...More data for this Ligand-Target Pair
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
IC50: 5.87E+4nMAssay Description:To gain insight into the selectivity of the synthetic compounds, nicotine, nicotine related alkaloids and nicotine metabolites for inhibition of othe...More data for this Ligand-Target Pair
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)
BDBM12341(CHEMBL178681 | CHEMBL359657 | US8609708, 1 | US860...)