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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM518688(US11116764, Compound 1 | US11253514, Compound 1 | ...)
Affinity DataKi:  2.04nMAssay Description:Table 2: Incubation conditions: Reactions were carried out in 50 mM Tris-HCl (pH 7.4) containing 10 mM MgCl2, 0.5 mM EDTA for 60 minutes at 37° C. Th...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM518688(US11116764, Compound 1 | US11253514, Compound 1 | ...)
Affinity DataKi:  2.04nMAssay Description:Example 2: Determination of Ki Value at 5-HT6 ReceptorCompound was tested at MDS pharma services and Novascreen according to the following procedures...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM518688(US11116764, Compound 1 | US11253514, Compound 1 | ...)
Affinity DataKi:  2.04nMAssay Description:Compound was tested at MDS pharma services and Novascreen according to the following procedures.Materials and Methods:Receptor source: Human recombin...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM518688(US11116764, Compound 1 | US11253514, Compound 1 | ...)
Affinity DataKi:  377nMAssay Description:Example 3: Determination of Ki Value at 5-HT2A ReceptorCompound was tested according to the following procedures.Materials and Methods:Receptor sourc...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM518688(US11116764, Compound 1 | US11253514, Compound 1 | ...)
Affinity DataKi:  2.51E+3nMAssay Description:Compound was tested according to the following procedures.Materials and Methods:Receptor source: Recombinant mammalian cellsRadioligand: [3H]-Ketanse...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Suven Life Sciences

US Patent
LigandPNGBDBM518688(US11116764, Compound 1 | US11253514, Compound 1 | ...)
Affinity DataKi:  2.51E+3nMAssay Description:Table 3: Incubation conditions: Reactions were carried out in 67 mM Tris-HCl (pH 7.4) for 4 hours at 37° C. The reaction was terminated by rapid vacu...More data for this Ligand-Target Pair
In DepthDetails US Patent