Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 11 hits in this display
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
IC50: 1.20E+3nMAssay Description:Inhibition of HDAC8 (unknown origin) using RHK(Ac)K(Ac) fluorogenic acetylated peptide substrate by fluorometric assayMore data for this Ligand-Target Pair
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
IC50: 2.70E+4nMAssay Description:Inhibition of HDAC5 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC fluorogenic acetylated peptide substrate by fluorometric assayMore data for this Ligand-Target Pair
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
IC50: 3.40E+4nMAssay Description:Inhibition of HDAC9 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC fluorogenic acetylated peptide substrate by fluorometric assayMore data for this Ligand-Target Pair
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
IC50: 4.90E+4nMAssay Description:Inhibition of HDAC7 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC fluorogenic acetylated peptide substrate by fluorometric assayMore data for this Ligand-Target Pair
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
IC50: 6.40E+4nMAssay Description:Inhibition of HDAC4 (unknown origin) using Boc-Lys(trifluoroacetyl)-AMC fluorogenic acetylated peptide substrate by fluorometric assayMore data for this Ligand-Target Pair
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
IC50: 6.79E+4nMAssay Description:To identify potential MBL inhibitors, the relative change in the formation of hydrolyzed nitrocefin between treated and untreated VIM2 was determined...More data for this Ligand-Target Pair
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)
BDBM50014161(CHEMBL3260858 | US11491146, Compound 5)