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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 27 hits in this display   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  93nMAssay Description:Binding affinity recombinant human BRD4 BD1 (42 to 168 residues) expressed in Escherichia coli BL21(DE3) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  96nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [49-170](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  96nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 2 [91-163](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  729nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 2 [91-163](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  729nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  742nMAssay Description:Binding affinity BRD2 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.17E+3nMAssay Description:Binding affinity human BRD4 BD2 incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4 [342-460](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.17E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 4 [342-460](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.17E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 2 [364-436](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.35E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 2 [364-436](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.35E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.38E+3nMAssay Description:Binding affinity BRD2 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3 [326-398](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.94E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [326-398](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.94E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.95E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.95E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  1.99E+3nMAssay Description:Binding affinity BRDT BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.02E+3nMAssay Description:Binding affinity BRD3 BD2 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3 [51-123](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.08E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3 [51-123](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.08E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.10E+3nMAssay Description:Binding affinity BRD3 BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain testis-specific protein [22-138](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.19E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain testis-specific protein [22-138](Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.19E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Md Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50:  2.22E+3nMAssay Description:Binding affinity BRDT BD1 (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50: >1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity CBP (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Board of Regents, The University of Texas System

US Patent
LigandPNGBDBM518799(US11117865, Compound ZL0591)
Affinity DataIC50: >1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent