Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 56 hits in this display
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 1.09E+4nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 1.14E+4nMpH: 7.4Assay Description:Carbonic anhydrase activity was assayed by following the change in absorbance at 348 nm of 4-nitrophenylacetate (NPA) to 4-nitrophenylate ion over a ...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 1.19E+4nMpH: 7.4Assay Description:Carbonic anhydrase activity was assayed by following the change in absorbance at 348 nm of 4-nitrophenylacetate (NPA) to 4-nitrophenylate ion over a ...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 1.22E+4nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 1.30E+4nM ΔG°: -27.9kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 4.89E+4nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 5.51E+4nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 6.06E+5nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 7.14E+5nMAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 4.00E+6nM ΔG°: -13.7kJ/molepH: 7.4 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA-catalyzed CO2 hydration activity. Phenol red has been used as indic...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
Ki: 4.01E+6nMpH: 7.4Assay Description:Carbonic anhydrase activity was assayed by following the change in absorbance at 348 nm of 4-nitrophenylacetate (NPA) to 4-nitrophenylate ion over a ...More data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
IC50: 5.90E+4nMAssay Description:Antagonist activity at LuxP receptor in Vibrio harveyi MM32 assessed as inhibition of autoinducer2-mediated quorum sensing after 3 to 4 hrsMore data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
IC50: >1.00E+5nMAssay Description:Inhibition of biotin-labelled p53 binding to MDM2 (25 to 109 residues) (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
BDBM26188(α-CA inhibitor, 12 | 1,2-Dihydroxybenzene, XI...)
IC50: 1.23E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
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