TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human TAOK3 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human TAOK3 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of human wild type partial length TAOK3 (M1 to T316 residues) expressed in mammalian expression system by Kinomescan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human TAOK3 using MBP substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human TAO3 N47S mutant (1 to 411 residues) using myelin basic protein as substrate incubated for 40 mins in presence of [ga...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of TAO3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAOK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of TAOK3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 86nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 0.220nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 86nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 210nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Binding affinity to TAOK3More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 310nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 5.00E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 720nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 4.60E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 490nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 210nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 390nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.40E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 590nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 99nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 2.20E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO3(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for TAOK3 kinase domainMore data for this Ligand-Target Pair