Affinity DataKi: 0.0110nMAssay Description:Tight binding inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 15 mins prior...More data for this Ligand-Target Pair
Affinity DataKi: 0.0110nM ΔG°: -62.5kJ/molepH: 7.4 T: 2°CAssay Description:Enzymatic assays were performed in the following reaction buffer: 50 mM HEPES, pH 7.4 containing 500 μg/ml bovine serum albumin. Enzyme activiti...More data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0610nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of recombinant matriptase (unknown origin) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hydrobromideMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.0880nMAssay Description:Tight binding inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 15 mins prior...More data for this Ligand-Target Pair
Affinity DataKi: 0.0880nM ΔG°: -57.4kJ/molepH: 7.4 T: 2°CAssay Description:Enzymatic assays were performed in the following reaction buffer: 50 mM HEPES, pH 7.4 containing 500 μg/ml bovine serum albumin. Enzyme activiti...More data for this Ligand-Target Pair
Affinity DataKi: 0.0920nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged matriptase catalytic domain expressed in Escherichia coli preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged matriptase catalytic domain expressed in Escherichia coli preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged matriptase catalytic domain expressed in Escherichia coli preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged matriptase catalytic domain expressed in Escherichia coli preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged matriptase catalytic domain expressed in Escherichia coli preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged matriptase catalytic domain expressed in Escherichia coli preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Compound was tested for inhibition of Matriptase from human breast cancer cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of recombinant matriptase (unknown origin) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hydrobromideMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of matriptase (unknown origin) using Boc-QAR-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of recombinant human matriptase preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tight binding inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 15 mins prior...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nM ΔG°: -50.5kJ/molepH: 7.4 T: 2°CAssay Description:Enzymatic assays were performed in the following reaction buffer: 50 mM HEPES, pH 7.4 containing 500 μg/ml bovine serum albumin. Enzyme activiti...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition assay using matriptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair