Report error Found 12 Enz. Inhib. hit(s) with Target = 'Urease subunit alpha/beta'
Affinity DataKi: 170nM ΔG°: -39.3kJ/mole IC50: 1.80E+3nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 1.75E+4nM ΔG°: -27.6kJ/mole IC50: 1.12E+5nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nM ΔG°: -27.5kJ/mole IC50: 6.00E+4nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+4nM ΔG°: -27.1kJ/mole IC50: 6.00E+4nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nM ΔG°: -26.7kJ/mole IC50: 8.00E+4nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+4nM ΔG°: -25.7kJ/mole IC50: 1.50E+5nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nM ΔG°: -25.3kJ/mole IC50: 1.23E+5nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+5nM ΔG°: -22.8kJ/mole IC50: 4.85E+5nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 1.35E+5nM ΔG°: -22.5kJ/mole IC50: 4.50E+5nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 2.15E+5nM ΔG°: -21.3kJ/mole IC50: 6.00E+5nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+5nM ΔG°: -20.1kJ/mole IC50: 1.10E+6nMpH: 7.0 T: 30°CAssay Description:Progress curves were obtained by initiation of urease reaction with addition of purified enzyme into assay mixtures containing increasing concentrati...More data for this Ligand-Target Pair
TargetUrease subunit alpha/beta(Helicobacter pylori (strain ATCC 700392 / 26695) (...)
Jishou University
Curated by ChEMBL
Jishou University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of Helicobacter pylori ATCC 43504 urease assessed as reduction in ammonia production preincubated for 1.5 hrs under cell free condition by...More data for this Ligand-Target Pair