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Found 39 Enz. Inhib. hit(s) with Target = 'Oxa40'
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227598(Penem 1)
Affinity DataKi:  30nM IC50:  150nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227599(Penem 3)
Affinity DataKi:  150nM IC50:  160nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92463(Imipenem)
Affinity DataKi:  3.20E+3nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50140672((2S,5R,6R)-6-Hydroxymethyl-3,3-dimethyl-7-oxo-4-th...)
Affinity DataKi:  3.00E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92461(Beta-lactam compound, 4)
Affinity DataKi:  4.20E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92464(Carbenicillin)
Affinity DataKi:  7.80E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50140671((2S,5R,6S)-6-Hydroxymethyl-3,3-dimethyl-7-oxo-4-th...)
Affinity DataKi:  8.30E+4nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM92462(Beta-lactam compound, 3)
Affinity DataKi:  4.04E+5nMAssay Description:Beta-lactam compounds were assessed as competitive inhibitors using nitrocefin as a reporter substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98796(US8487093, 184)
Affinity DataIC50:  360nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98792(US8487093, 180)
Affinity DataIC50:  530nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98800(US8487093, 190)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98787(US8487093, 170)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50315411(4,7-Dichloro-1-benzothien-2-yl sulfonylaminomethyl...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Acinetobacter baumannii beta-lactamase OXA40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347181(CHEMBL1795564)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347181(CHEMBL1795564)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98824(US8487093, 222)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347184(CHEMBL1795567)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98791(US8487093, 178)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50447649(CHEMBL3112746)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347185(CHEMBL1795568)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347183(CHEMBL1795566)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347188(CHEMBL1795571)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50447647(CHEMBL3112752)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347189(CHEMBL1795572)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98735(US8487093, 80)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50447651(CHEMBL3112741)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50447650(CHEMBL3112742)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98734(US8487093, 78)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98737(US8487093, 82)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98742(US8487093, 90)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50447648(CHEMBL3112750)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98755(US8487093, 116)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM98764(US8487093, 132)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50447652(CHEMBL3112756)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of beta-lactamase Oxa40 in Acinetobacter baumannii assessed as inhibition of hydrolysis of nitrocefinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347187(CHEMBL1795570)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347186(CHEMBL1795569)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347182(CHEMBL1795565)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347180(CHEMBL1795563)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM50347188(CHEMBL1795571)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Acinetobacter baumannii beta lactamase OXA-40More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed