Query String: Muscimol
Muscimol BDBM50052792 CHEBI:7035
CAS_2763-96-4 NSC_4266 BDBM85713 Muscimol
Pantherine BDBM23183 Agarin Muscimol 5-(aminomethyl)-1,2-oxazol-3-ol CHEMBL273481
- Melikian, A; Schlewer, G; Chambon, JP; Wermuth, CG Condensation of muscimol or thiomuscimol with aminopyridazines yields GABA-A antagonists. J Med Chem 35: 4092-7 (1992)
- Herschel, M; Baldessarini, RJ Evidence for two types of binding of 3H-gaba and 3H-muscimol in rat cerebral cortex and cerebellum. Life Sci 24: 1849-54 (1979)
- Petersen, JG; Bergmann, R; Møller, HA; Jørgensen, CG; Nielsen, B; Kehler, J; Frydenvang, K; Kristensen, J; Balle, T; Jensen, AA; Kristiansen, U; Frølund, B Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as¿-aminobutyric acid(a) receptor agonists. J Med Chem 56: 993-1006 (2013)
- Williams, M; Risley, EA Characterization of the binding of [3H]muscimol, a potent gamma-aminobutyric acid agonist, to rat brain synaptosomal membranes using a filtration assay. J Neurochem 32: 713-8 (1979)
- Ray2010 Assay 70 muscimol cortex .
- ChEBML_219116 Inhibition of [3H]muscimol binding to GABA-A of rat cerebellum
- ChEBML_68589 Inhibition of [3H]muscimol binding to Gamma-aminobutyric acid (GABA-A) receptor
- ChEMBL_514066 (CHEMBL979089) Displacement of [3H]Muscimol from GABAAalpha6 receptor in Sprague-Dawley rat brain cerebellum membrane
- ChEMBL_1881819 (CHEMBL4383318) Displacement of [3H]muscimol from recombinant human GABAalpha1beta2gamma2 measured after 120 mins by scintillation counting method
- ChEMBL_2186850 (CHEMBL5098932) Displacement of [3H]-muscimol from human GABAA alpha1beta3gamma2 stably expressed in Ltk cells assessed as inhibition constant by liquid scintillation counting method
- ChEMBL_1724104 (CHEMBL4139382) Displacement of [3H]muscimol from human GABAA receptor alpha1beta3gamma2 expressed in HEK293 TetR cell membranes after 1 hr by liquid scintillation counting method
- ChEMBL_1767464 (CHEMBL4219576) Agonist activity at GABAA receptor in Sprague-Dawley rat forebrain membranes assessed as enhancement of [3H]muscimol binding after 2 hrs by radiometric analysis
- ChEMBL_2032691 (CHEMBL4686849) Positive allosteric modulation of GABAA alpha1beta3gamma2L in HEK cell plasma membrane assessed as increase in [3H]muscimol binding measured after 10 mins by liquid scintillation counting method
- ChEMBL_2032692 (CHEMBL4686850) Positive allosteric modulation of GABAA alpha1beta3 in HEK cell plasma membrane assessed as increase in [3H]muscimol binding measured after 10 mins by liquid scintillation counting method