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Found 6 of ic50 for monomerid = 515341
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Acerta Pharma

US Patent
LigandPNGBDBM515341(US11110088, Compound Table 1.15)
Affinity DataIC50:  2.20nMAssay Description:BTK enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.BTK enzyme (H...More data for this Ligand-Target Pair
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TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Acerta Pharma

US Patent
LigandPNGBDBM515341(US11110088, Compound Table 1.15)
Affinity DataIC50:  3.40nMAssay Description:TEC enzyme (Millipore #14-801M), is diluted to 2 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.1% NaN3, 1 mM DTT, 2 mM MnCl2, pH ...More data for this Ligand-Target Pair
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TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
Acerta Pharma

US Patent
LigandPNGBDBM515341(US11110088, Compound Table 1.15)
Affinity DataIC50:  3.5nMAssay Description:BMX enzyme (Millipore #14-499M), is diluted to 0.5 U/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.1% NaN3, 1 mM DTT, 2 mM MnCl2, p...More data for this Ligand-Target Pair
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TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Acerta Pharma

US Patent
LigandPNGBDBM515341(US11110088, Compound Table 1.15)
Affinity DataIC50:  4.70nMAssay Description:TXK enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.TXK enzyme (M...More data for this Ligand-Target Pair
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TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Acerta Pharma

US Patent
LigandPNGBDBM515341(US11110088, Compound Table 1.15)
Affinity DataIC50: >1.00E+3nMAssay Description:ITK enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.ITK enzyme (M...More data for this Ligand-Target Pair
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TargetEpidermal growth factor receptor(Homo sapiens (Human))
Acerta Pharma

US Patent
LigandPNGBDBM515341(US11110088, Compound Table 1.15)
Affinity DataIC50: >1.00E+3nMAssay Description:EGFR enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.EGFR enzyme ...More data for this Ligand-Target Pair
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In DepthDetails US Patent