TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.00260nMAssay Description:Binding affinity of the compound against Opioid receptor delta 1 using [3H]-DT in rat brain synaptosomes was determinedMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Inhibition of [3H]-DADLE binding to opioid receptor delta in P2 membrane preparation of rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Binding affinity against opioid receptor delta in rats by displacing [3H]-DPDPEMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]deltorphin II from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Inhibition of [3H]-naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of [3H]- DPDPE binding to delta opioid receptor of guinea pig brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University
Curated by ChEMBL
Tohoku Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 147nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 147nMAssay Description:Opioid receptor mu 1 binding affinity by displacement of radioligand [3H][DAla,MePhe,Gly-ol]enkephalin (DAGO) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 147nMAssay Description:Displacement of [3H]-DAGO (1.28 nM) from Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 262nMAssay Description:Inhibition of [3H]- ]DAMGO binding to opioid receptor mu from rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 272nMAssay Description:Binding affinity against opioid receptor mu in rats by displacing [3H]-DAGOMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 272nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 314nMAssay Description:Binding affinity of the compound against Opioid receptor mu 1 using [3H]-DAMGO in rat brain synaptosomes was determinedMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 387nMAssay Description:Inhibition of [3H]DAGO binding to trat brain opioid receptor mu in P2 membraneMore data for this Ligand-Target Pair
Affinity DataKi: 677nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of guinea pig brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of [3H]-naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
Affinity DataKi: 1.98E+3nMAssay Description:Displacement of [3H]-DAGO from Opioid receptor mu 1 of adult male mouse brain.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute of Environmental Health Sciences
Curated by ChEMBL
National Institute of Environmental Health Sciences
Curated by ChEMBL
Affinity DataKi: 3.93E+3nMAssay Description:Tested for binding affinity against mu opioid receptor fby displacing [3H]- DAMGO radioligand from rat brain membrane preparationsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Eastern Michigan University
Curated by ChEMBL
Eastern Michigan University
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]- U 69593 from Opioid receptor kappa 1 of guinea pig brainMore data for this Ligand-Target Pair