Affinity DataKd: 4.30nMpH: 5.5Assay Description:Saturation binding of mutant human Adenosine A2A receptor (H250N) at pH 5.5More data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:Displacement of [3H]4-[2-[7-amino-2-(2-furyl)-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-yl-amino]ethylphenol from wild type human adenosine A2a receptor ...More data for this Ligand-Target Pair
Affinity DataKd: 7.60nMAssay Description:Kd in saturation experiments using [3H]CGS-21680 at H250N mutant receptor in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 7.60nMpH: 6.8Assay Description:Saturation binding of human Adenosine A2A receptor (H250N) at pH 6.8More data for this Ligand-Target Pair
Affinity DataKd: 12nMpH: 7.5Assay Description:Saturation binding of human Adenosine A2A receptor H250N at pH 7.5More data for this Ligand-Target Pair
Affinity DataKd: 22nMpH: 5.5Assay Description:Saturation binding characteristics of wild type human Adenosine A2A receptor at pH 5.5More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Kd in saturation experiments using [3H]CGS-21680 at V84L mutant receptor in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 36nMpH: 6.8Assay Description:Saturation binding of wild type human Adenosine A2A receptor at pH 6.8More data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Kd in saturation experiments using [3H]CGS-21680 at WT receptor in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 74nMpH: 7.5Assay Description:Saturation binding characteristics of wild type human Adenosine A2A receptor at pH 7.5More data for this Ligand-Target Pair
Affinity DataKd: 99nMpH: 8.4Assay Description:Saturation binding of human Adenosine A2A receptor H250N at pH 8.4More data for this Ligand-Target Pair
Affinity DataKd: 632nMpH: 8.4Assay Description:Saturation binding of wild type human Adenosine A2A receptor at pH 8.4More data for this Ligand-Target Pair