Affinity DataKd: 0.00560nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.0200nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.0210nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.0210nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: <0.200nMAssay Description:Binding affinity to His6-tagged recombinant human ROCK2 by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Affinity DataKd: <0.200nMAssay Description:Binding affinity to His6-tagged recombinant human ROCK2 by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.700nMAssay Description:Displacement of fluorescent-ARC-1042 from His6-tagged recombinant human ROCK2 by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Affinity DataKd: <1nMAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: <1nMAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding affinity to ROCK2 (unknown origin) incubated for 1 hr by qPCR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Displacement of fluorescent-ARC-1042 from His6-tagged recombinant human ROCK2 by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Affinity DataKd: <3nMAssay Description:Displacement of ARC583 from ROCK2More data for this Ligand-Target Pair
Affinity DataKd: <3nMAssay Description:Displacement of ARC583 from ROCK2More data for this Ligand-Target Pair
Affinity DataKd: 3.80nMAssay Description:Displacement of ARC583 from ROCK2More data for this Ligand-Target Pair
Affinity DataKd: 6.40nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged ROCK2 (unknown origin) (1 to 553 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair
Affinity DataKd: 23nMAssay Description:Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged ROCK2 (unknown origin) (1 to 553 residues) expressed in baculovirus infect...More data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Inhibition of ROCK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 31nMpH: 7.5 T: 2°CAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Displacement of ARC583 from ROCK2More data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 46nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 65nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 71nMAssay Description:Binding affinity to ROCK2More data for this Ligand-Target Pair
Affinity DataKd: 71nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 78nMAssay Description:Displacement of fluorescent-ARC-1063 from His6-tagged recombinant human ROCK2 by luminescence intensity assayMore data for this Ligand-Target Pair
Affinity DataKd: 89.7nMpH: 7.5 T: 2°CAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: 119nMAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding affinity to ROCK2More data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 177nMAssay Description:Displacement of ARC583 from ROCK2More data for this Ligand-Target Pair
Affinity DataKd: 187nMAssay Description:The assay is based on the kinase-bound labeled fluorescent probe can be displaced by competitive inhibitors, which can be registered by measurement o...More data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to wild-type partial length human ROCK2 (M1 to T431 residues) expressed in mammalian expression system by Kinomescan assayMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to wild-type partial length human ROCK2 (M1 to T431 residues) expressed in mammalian expression system by Kinomescan assayMore data for this Ligand-Target Pair
Affinity DataKd: 230nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding constant for ROCK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 280nMAssay Description:Compounds were tested using an 11-point curve with 3-fold serial dilutions. IC50 determinations were made using an ATP concentration of 10 uM. The hi...More data for this Ligand-Target Pair
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