Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50004309
TargetNonstructural protein 3(Zika virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212337(CHEMBL5267698)
Affinity DataKi:  1.70nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212337(CHEMBL5267698)
Affinity DataKi:  69nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50030459(CHEMBL3344321)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212336(CHEMBL5282745)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212339(CHEMBL4173093)
Affinity DataKi:  3.06E+3nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212340(CHEMBL5276951)
Affinity DataKi:  4.47E+3nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50026808(CHEMBL2440341)
Affinity DataKi:  9.25E+4nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50030459(CHEMBL3344321)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212341(CHEMBL5287718)
Affinity DataKi:  5.00E+5nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50030459(CHEMBL3344321)
Affinity DataKi: >5.00E+5nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM35491(Benzoic acid 5-amino-1-(4-methoxy-benzenesulfonyl)...)
Affinity DataIC50:  105nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212335(CHEMBL5275144)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50567466(CHEMBL4862682)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50218663(CHEMBL5269219)
Affinity DataIC50:  440nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50108877((3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone |...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50567466(CHEMBL4862682)
Affinity DataIC50:  710nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50241035(1-[(1R,2R,4S,5S)-5-carbamimidamido-2,4-bis(2,4-dic...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50030456(CHEMBL3344319)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50212338(CHEMBL5290934)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50490541(CHEMBL1457139)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50490541(CHEMBL1457139)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50218663(CHEMBL5269219)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against cell free dihydrofolate redutase (DHFR) from Mycobacterium lufuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50468907(CHEMBL549740)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Charles University Prague

Curated by ChEMBL
LigandPNGBDBM50468907(CHEMBL549740)
Affinity DataKd:  4.00E+4nMAssay Description:Inhibitory activity against cell free dihydrofolate reductase (DHFR) from Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed