Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50004977
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128175(1,1,1-Trifluoro-3-{[3-(3-isopropyl-phenoxy)-phenyl...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128154(1,1,1-Trifluoro-3-{[3-(1,1,2,2-tetrafluoro-ethoxy)...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128164(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-chlo...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128141(1,1,1-Trifluoro-3-{[3-(4-fluoro-phenoxy)-phenyl]-[...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128135(3-((3-(2,3-dichlorophenoxy)phenyl)(3-(1,1,2,2-tetr...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128146(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(3-ethy...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128169(1,1,1-Trifluoro-3-{[3-(4-fluoro-3-methyl-phenoxy)-...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128185(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(3-ethy...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128167(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(3,4-di...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128152(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(3-tert...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128166(1,1,1-Trifluoro-3-{[3-(1,1,2,2-tetrafluoro-ethoxy)...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128143(1,1,1-Trifluoro-3-[[3-(1,1,2,2-tetrafluoro-ethoxy)...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128168(1,1,1-Trifluoro-3-[[3-(1,1,2,2-tetrafluoro-ethoxy)...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128162(1,1,1-Trifluoro-3-{[3-(1,1,2,2-tetrafluoro-ethoxy)...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128148(1,1,1-Trifluoro-3-{[3-(3-fluoro-2-nitro-phenoxy)-p...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128173(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-chlo...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128184(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(3-(dim...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128133(1,1,1-Trifluoro-3-{[3-(4-isopropyl-3-methyl-phenox...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128132(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(3,5-di...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128155(1,1,1-Trifluoro-3-{[3-(4-propyl-phenoxy)-phenyl]-[...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128145(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-chlo...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128182(1,1,1-Trifluoro-3-{[3-(3-fluoro-phenoxy)-phenyl]-[...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128159(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(2-chlo...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128171(1,1,1-Trifluoro-3-{[3-(1,1,2,2-tetrafluoro-ethoxy)...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128181(1,1,1-Trifluoro-3-{[3-(4-propoxy-phenoxy)-phenyl]-...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128174(1,1,1-Trifluoro-3-{[3-(4-nitro-phenoxy)-phenyl]-[3...)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128151(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-amin...)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128130(1,1,1-Trifluoro-3-{[3-(3-methoxy-phenoxy)-phenyl]-...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128144(3-((3-(1,1,2,2-tetrafluoroethoxy)benzyl)(3-(4-benz...)
Affinity DataIC50:  2.40E+6nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholesteryl ester transfer protein(Homo sapiens (Human))TBA
LigandPNGBDBM50128179(3-((3-(biphenyl-4-yloxy)phenyl)(3-(1,1,2,2-tetrafl...)
Affinity DataIC50:  2.50E+6nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails Article