Found 5 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50128181'
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia
Curated by ChEMBL
Universidade Federal Da Bahia
Curated by ChEMBL
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia
Curated by ChEMBL
Universidade Federal Da Bahia
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Compound was tested in vitro for inhibitory activity against recombinant human cholesteryl ester transfer protein in bufferMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Oryctolagus cuniculus)
Al-Zaytoonah Private University Of Jordan
Curated by ChEMBL
Al-Zaytoonah Private University Of Jordan
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia
Curated by ChEMBL
Universidade Federal Da Bahia
Curated by ChEMBL
Affinity DataIC50: 3.42E+4nMAssay Description:Compound was tested in vitro for inhibitory activity against recombinant human cholesteryl ester transfer protein in human serumMore data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia
Curated by ChEMBL
Universidade Federal Da Bahia
Curated by ChEMBL
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of CETP (unknown origin)-mediated [3H]cholesteryl ester transfer from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair