TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 104nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 114nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 133nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 142nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 199nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 203nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 231nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 295nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 331nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 364nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 367nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 430nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 717nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 828nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 846nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Heinrich Heine University Duesseldorf
Curated by ChEMBL
Affinity DataKi: 941nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair