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Found 19 Enz. Inhib. hit(s) with all data for entry = 50018632
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50196467(3-(4-chlorobenzyl)-N-(3-(2-ethylpiperidin-1-yl)pro...)
Affinity DataIC50:  100nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50148172(CHEMBL251949 | KYS-05042 | N-(4-(4-fluorophenylsul...)
Affinity DataIC50:  200nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50148180(2-(3-Phenyl-2-piperidin-1-yl-3,4-dihydro-quinazoli...)
Affinity DataIC50:  250nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50117922((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...)
Affinity DataIC50:  840nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50148175(CHEMBL114695 | KYS-05001 | N-Benzyl-2-(3-phenyl-2-...)
Affinity DataIC50:  900nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192101(2-(3-ethyl-2-(piperidin-1-yl)-3,4-dihydroquinazoli...)
Affinity DataIC50:  960nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197630(CHEMBL227905 | N-((3-(2-(trifluoromethyl)phenyl)is...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197623(3-(4-chlorobenzyl)-N-(3-(4-methylpiperidin-1-yl)pr...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197622(3-(4-chlorobenzyl)-4-oxo-N-(3-(pyrrolidin-1-yl)pro...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197621(3-(4-chlorobenzyl)-N-(3-(azepan-1-yl)propyl)-4-oxo...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197624(2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197633(2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-...)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197632(CHEMBL436133 | N-((3-(2-methoxyphenyl)isoxazol-5-y...)
Affinity DataIC50:  2.04E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197628(3-(4-chlorobenzyl)-4-oxo-N-(3-(piperidin-1-yl)prop...)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197625(3-(4-chlorobenzyl)-N-(3-(4-ethylpiperazin-1-yl)pro...)
Affinity DataIC50:  2.53E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197629(3-(4-chlorobenzyl)-N-(3-(benzyl(methyl)amino)propy...)
Affinity DataIC50:  4.69E+3nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197626(3-(4-chlorobenzyl)-N-(2-(butyl(methyl)amino)ethyl)...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197627(3-(4-chlorobenzyl)-7-(1-methylpiperazine-4-carbony...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50197631(3-(4-chlorobenzyl)-N-(2-(dimethylamino)ethyl)-4-ox...)
Affinity DataIC50:  5.35E+4nMAssay Description:Inhibition of alpha1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed