Affinity DataKi: 0.170nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-pentazocine from guinea pig sigma1 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 10.9nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 13.2nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 13.4nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 13.6nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 13.8nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 14.2nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 15.1nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 15.1nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 17.7nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 17.8nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 18.2nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 18.5nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 19.6nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 20.9nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 21.4nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 24.2nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 24.9nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 27.1nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 27.7nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 31.7nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 34.4nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 35.2nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 37.9nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 54.5nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 55.3nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 57.6nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 59.2nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 64.8nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 70.5nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Binding affinity to human D4 receptor transfected in human HEK293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Binding affinity to human D4 receptor transfected in human HEK293 cells by gamma-countingMore data for this Ligand-Target Pair