Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50034491
Affinity DataIC50: 0.0820nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.220nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.450nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.670nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 990nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+3nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.33E+3nMAssay Description:Displacement of radiolabeled FK33-824 from mu opioid receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Astrazeneca Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair