Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50040974
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant Btk after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Irreversible inhibition of EGFRMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Btk in human Ramos cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of RSK2 transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of EGF-induced autophosphorylation of EGFR in human A431 cellsMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Covalution Pharma
Curated by ChEMBL
Covalution Pharma
Curated by ChEMBL
TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Covalution Pharma
Curated by ChEMBL
Covalution Pharma
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of GST-tagged EGFR expressed in sf9 cells by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Inhibition of recombinant FGFR1More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK2 transfected in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of GST-tagged Plk1 using recombinant protein X as a substrate containing threonine residuesMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of GST-tagged ErbB2 expressed in sf9 cells by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of GST-tagged ErbB4 expressed in sf9 cells by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 149nMAssay Description:Inhibition of human AKT1 using biotinylated GSKalpha peptide (SGRARTSSFA) as a substrate after 1 hrMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 7(Human)
Covalution Pharma
Curated by ChEMBL
Covalution Pharma
Curated by ChEMBL
Affinity DataIC50: 313nMAssay Description:Inhibition of human AKT1 using biotinylated GSKalpha peptide (SGRARTSSFA) as a substrate after 1 hrMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Human)
Covalution Pharma
Curated by ChEMBL
Covalution Pharma
Curated by ChEMBL
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of MKK4More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of chicken c-Src using IYGEFKKK peptide as a substrate and [32P]ATP by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of chicken c-SrcMore data for this Ligand-Target Pair
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of chicken c-SrcMore data for this Ligand-Target Pair
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of chicken c-SrcMore data for this Ligand-Target Pair
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of chicken c-SrcMore data for this Ligand-Target Pair