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Found 18 Enz. Inhib. hit(s) with all data for entry = 50048347
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataIC50:  0.900nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colon in presence of phentolamine (10 uM), desmethylimipramine (0.5 uM) and hydrocortisone (30 uM)More data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212980(CHEMBL553039 | SR-58997A)
Affinity DataIC50:  1.10nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colon in presence of phentolamine (10 uM), desmethylimipramine (0.5 uM) and hydrocortisone (30 uM)More data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataIC50:  3.5nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colon in presence of phentolamine (10 uM), desmethylimipramine (0.5 uM) and hydrocortisone (30 uM)More data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212979(CHEMBL543333)
Affinity DataIC50:  21nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colonMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataIC50:  47nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colonMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212978(CHEMBL541542)
Affinity DataIC50:  90nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colonMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212978(CHEMBL541542)
Affinity DataIC50:  185nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212980(CHEMBL553039 | SR-58997A)
Affinity DataIC50:  319nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212979(CHEMBL543333)
Affinity DataIC50:  350nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataIC50:  480nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataIC50:  1.20E+3nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataIC50:  1.20E+3nMAssay Description:Beta-adrenergic agonistic activity in rat uterus preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212977(AMIBEGRON HYDROCHLORIDE | Amibegron HCl | SR-58611...)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212980(CHEMBL553039 | SR-58997A)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212979(CHEMBL543333)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-1/Beta-2/Beta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212978(CHEMBL541542)
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
In DepthDetails