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Found
1
Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase type 2' and Ligand = 'BDBM642875'
Target
11-beta-hydroxysteroid dehydrogenase type 2
(Homo sapiens (Human))
Ardelyx
US Patent
Ligand
BDBM642875
((2S,4aS,6aS,6bR,8aR,9S,10S,12aS,12bR,14bR)-2,4a,6a...)
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Affinity Data
IC50: 10nM
Assay Description:
Human descending colon epithelial stem cells were cultured as 3D organoids in accordance with Sato et al Gastroenterology. 2011 November; 141(5): 176...
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Target Info
Reactome pathway
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Ligand Info
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Details
US Patent
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