Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM110163'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
North-West University

Curated by ChEMBL
LigandPNGBDBM110163(8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d))
Affinity DataKi:  139nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat brain cortical membranes in absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
North-West University

Curated by ChEMBL
LigandPNGBDBM110163(8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d))
Affinity DataKi:  164nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat whole brain membranes in absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
North-West University

Curated by ChEMBL
LigandPNGBDBM110163(8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d))
Affinity DataKi:  164nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Isf College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM110163(8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d))
Affinity DataKi:  164nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
North-West University

Curated by ChEMBL
LigandPNGBDBM110163(8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d))
Affinity DataKi:  209nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat whole brain membranes in presence of 0.1 mM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
North-West University

Curated by ChEMBL
LigandPNGBDBM110163(8-(3-Phenylpropyl)-1,3,7-triethylxanthine (9d))
Affinity DataKi:  258nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor in Sprague-Dawley rat brain cortical membranes in presence of 0.1 mM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed