Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3' and Ligand = 'BDBM50604885'
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataKi: >4.00E+5nMAssay Description:Binding affinity to recombinant human BRD3 BD2 (306-417 residues) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Yancheng Teachers University
Curated by ChEMBL
Yancheng Teachers University
Curated by ChEMBL
Affinity DataKi: >4.00E+5nMAssay Description:Binding affinity to recombinant human BRD3 BD1 (24-144 residues) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair