Affinity DataKi: 31nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inverse agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inverse agonist activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 31.2nMAssay Description:Binding affinity to cannabinoid CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 31.2nMAssay Description:Binding affinity for human cannabinoid receptor 2 was determined by using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 31.2nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
Affinity DataKi: 35.8nMAssay Description:Binding assay with hCB1 and hCB2 receptors.More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 expressed in CHO cells after 90 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at cannabinoid CB2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Inverse agonist activity at C-terminally prolink-tagged mouse CB2 receptor expressed in CHOK1 cells harboring beta-galactosidase enzyme fused beta-ar...More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Inverse agonist activity at mouse CB2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-mediated cAMP accumulation after 5 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 167nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 90 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 76.6nMAssay Description:Agonist activity at human CB2 receptor expressed CHO cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.15E+3nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
Affinity DataEC50: 603nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in Sf9 cells coexpressing Galpha i2 assessed as Galpha GTPase activity using [gamma-33P]GTP ...More data for this Ligand-Target Pair